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SMS - Brevets
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2011
Methods for the preparation of (3S,3S')4,4'Disulfanediylbis (3-Aminobutane 1-sulfonic acid) WO2012045849, 12/04/2010. Balavoine F.; Madec J.; Schneider J.M.; Coquerel G.; Couvrat N.; Cartigny Y.; Petit M.N.
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2010
Compositions pharmaceutiques du 6-oxo-6,7,8,9,10,11-hexahydrocyclohepta 3-yl sulfamate. PCT/FR2010/000117, 2010. Mondoly, N.; Poirot, B.; Brochard, A.; Richard, J.; Delahaye, D.; Diolez, C.; Rolland, A.; Diancourt, F.; Coquerel, G.; Martins, D.; Linol, J.; Houssin, O.; Petit, M.-N.; Potter, B. V. L.; Woo, L. W. L. Novel process for obtaining the crystalline form V of Agomelatine. WO/2010/015747, 11/02/2010, 2010.
Martins, D.; Coquerel, G.; Linol, J.; Langlois, P. Process for enantiomeric separation of racemic dihydro-1, 3, 5 triazines via preferential crystallization. WO2010109015 (A1), 2010-09-30, 2010. 4.
Helmreich, M.; Niesert, C.-P.; Cravo, D.; Coquerel, G.; Levilain, G.; Wacharine-Antar, s.; Cardinaël, P. Novel Polymorphic form of CHDMAPP, method of preparation thereof, and pharmaceutical composition comprising same. WO2010/029062 A1, 18.03.2010, 2010.
Descamps, G.; Amharar, Y.; Cartigny, Y.; Coquerel, G. New polymorph of 6-oxo-6, 7, 8, 9, 10, 11-hexahydrocyclohepta(c) chromen-3-yl sulfamate having specific particle size, is steroid sulfatase inhibitor, useful to treat cancer and hormone-dependent cancers e.g. breast cancer. FR2942225 (A1), 2010-08-20, 2010.
Delahaye, D.; Diolez, C.; Rolland, A.; Diancourt, F.; Brochard, A.; Mondoly, N.; Poirot, B.; Coquerel, G.; Martins, D.; Linol, J.; Potter, B. V. L.; Woo, L. W. L. New polymorphic form, crystalline dimethyl sulfoxide solvate and crystalline 1, 4-dioxane hemisolvate of 6-oxo-6, 7, 8, 9, 10, 11-hexahydrocyclohepta(c)chromen-3-yl sulfamate, are steroid sulfatase inhibitors, useful to treat cancer. FR2942226 (A1), 2010-08-20, 2010.
Delahaye, D.; Diolez, C.; Rolland, A.; Diancourt, F.; Brochard, A.; Mondoly, N.; Poirot, B.; Coquerel, G.; Martins, D.; Houssin, O.; Petit, M.-N. Novel Polymorphic form of CHDMAPP, method of preparation thereof, and pharmaseutical composition comprising same. WO2010/029062 A1, 18.03.2010, 2010.
Descamps, G.; Amharar, Y.; Cartigny, Y.; Coquerel, G. Novel process for obtaining the crystalline form V of Agomelatine. WO/2010/015747, 11/02/2010, 2010.
Martins, D.; Coquerel, G.; Linol, J.; Langlois, P. Compositions pharmaceutiques du 6-oxo-6,7,8,9,10,11-hexahydrocyclohepta 3-yl sulfamate. PCT/FR2010/000117, 2010. WO/2010/092260.
Mondoly, N.; Poirot, B.; Brochard, A.; Richard, J.; Delahaye, D.; Diolez, C.; Rolland, A.; Diancourt, F.; Coquerel, G.; Martins, D.; Linol, J.; Houssin, O.; Petit, M.-N.; Potter, B. V. L.; Woo, L. W. L. 
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2009
Novel crystalline form VI of agomelatine, method for preparing same and pharmaceutical compositions containing same. WO2009095555, 06/08/2009, 2009.
Coquerel, G.; Linol, J.; Le Pape, L.; Lecouvé, J.-P.Rimonabant N-methylpyrrolidone solvate, method for preparing same and pharmaceutical compositions containing same. WO2009053550, 30/04/2009, 2009.
Coquerel, G.; Fours, B. Rimonabant N, N-dimethylformamide solvate, and method for preparing same. WO2009053551, 30/04/2009, 2009.
Coquerel, G.; Fours, B. Rimonabant DMSO solvate, method for preparing same and pharmaceutical compositions containing same. WO2009053549, 30/04/2009, 2009.
Coquerel, G.; Fours, B. Rimonabant 2-methoxyethanol solvate and method for preparing same. WO2009053553, 30/04/2009, 2009.
Coquerel, G.; Fours, B. Rimonabant 1, 4-dioxane solvate, method for preparing same and pharmaceutical compositions containing same. WO2009053548, 30/04/2009, 2009.
Coquerel, G.; Fours, B. Isopropanol solvate of rimonabant, preparation method thereof and pharmaceutical compositions containing same. WO2009050354, 23/04/2009, 2009.
Coquerel, G.; Fours, B. 3-methylbutan-1-ol solvate of rimonabant, preparation method thereof and pharmaceutical compositions containing same. WO2009050353, 23/03/2009, 2009.
Coquerel, G.; Fours, B. Method for splitting omeprazole salts. WO 2009/027614 A2, 05.03.2009, 2009.
Coquerel, G.; Tauvel, G.; Petit, M.-N. Rimonabant monohydrate, process for the preparation thereof and pharmaceutical compositions containing same. US2009048449, 19/02/2009, 2009.
Coquerel, G.; Duplaa, H.; Fours, B.; Monnier, O.; Ochsenbein, P.
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2008
Cristalline phases of 5,6-Dichloro-2-(isopropylamino)-(1--L-Ribofuranosyl)-1H-Benzimidazole. PVMB-0386P1, 23-12-2008, 2008.
Coquerel, G.; Levilain, G.; Petit, M.-N.; Coste, S.Conglomerates of tenatoprazole potassium salts. WO2008081104(A2), 2008-07-10, 2008.
Cohen, A.; Schutze, F.; Charbit, S.; Bernad, S.; Tauvel, G.; Petit, M.-N.; Coquerel, G.
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2007
a crystalline form of the arginine salt of perindopril, process for preparing it, and pharmaceutical compositions comprising it. WO2007099217(A1), 2007-09-07, 2007.Coquerel, G.; Lefèbvre, L.; Souvie, J.-C.; Authouart, P.ss-crystalline form of perindopril arginine salt, method for making same, and pharmaceutical compositions containing same. WO2007099216(A2), 2007-09-07, 2007.
Coquerel, G.; Lefèbvre, L.; Souvie, J.-C.; Authouart, P. Novel crystalline V form of agomelatine, method of the preparation thereof and pharmaceutical compositions containing said form. WO2007015004, 08/02/2007, 2007.
Coquerel, G.; Linol, J.; Souvie, J.-C. Novel crystalline IV form of agomelatine, method of the preparation thereof and pharmaceutical compositions containing said form. WO 2007 015002, 08/02/2007, 2007.
Coquerel, G.; Linol, J.; Souvie, J.-C. Novel crystalline III form of agomelatine, method of the preparation thereof and pharmaceutical compositions containing said form. WO 2007 015003, 08/02/2007, 2007.
Coquerel, G.; Linol, J.; Souvie, J.-C.
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2006
Conglomérats de sels de potassium du ténatoprazole. FR N°06/10553, 04/12/2006, 2006.
Coquerel, G.; Tauvel, G.; Petit, M.-N. Forme cristalline du sel d'arginine du perindopril, son procédé de préparation et les compositions pharmaceutiques qui la contiennent. FR N°06/01748, 2006
Coquerel, G.; Lefèbvre, L.; Souvie, J.-C.; Authouart, P. Forme cristalline du sel d'arginine du perindopril, son procédé de préparation et les compositions pharmaceutiques qui la contiennent. FR N°06/01748, 2006
Coquerel, G.; Lefèbvre, L.; Souvie, J.-C.; Authouart, P. Le monohydrate de Rimonabant, son procédé de préparation et les compositions pharmaceutiques qui en contiennent. FR N°06/01253, 2006
Coquerel, G.; Fours, B. Polymorphic forms V of Agomelatine, its methods of preparation and its pharmaceutical compositions. FR N°05/08278, 2005
Coquerel, G.; Linol, J.; Souvie, J.-C.
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2005
Polymorphic forms IV of Agomelatine, its methods of preparation and its pharmaceutical compositions. FR N°05/08277, 2005.
Coquerel, G.; Linol, J.; Souvie, J.-C.Polymorphic forms III of Agomelatine, its methods of preparation and its pharmaceutical compositions. FR N°05/08276, 03/08/2005, 2005.
Coquerel, G.; Linol, J.; Souvie, J.-C. Phosphoantigen Salts of Organic Bases and Methods for their Crystallization. Purification by means of crystallization of some Pyrophosphate analogous antigen. US patent N°60/724,308, 06/10/2005, 2005.
Coquerel, G.; Aubin, E.
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2004
Polymorphic forms of Fasidotril, their methods of preparation and pharmatical compositions comprising them. 27/07/2004, 2004.
Capet, M.; Coquerel, G.; Danvy, D.; Lecomte, J.-M.; Petit, M.-N.; Schwartz, J. C. Modafinil Polymorphic forms. 19/02/2004, 2004.
Broquaire, M.; Courvoisier, L.; Mallet, F.; Coquerel, G.; Frydman, A.
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2003
Method for preparation of modafinil enantiomers and crystalline forms of optical enantiomers of modafinil. French Patent N°02/04036, 20/12/2003, 2003.
Neckebrock, O.; Courvoisier, L.; Graf, S.; Serrure, G.; Coquerel, G.; Rose, S.; Besselièvre, C.
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2002
Polymorphic forms and solvates of -Modafinil. US Patent N°60/402064, 08/08/2002, 2002. Broquaire, M.; Courvoisier, L.; Branger-Zagouri, C.; Rose, S.; Coquerel, G.
Formes polymorphes du Fasidotril, leur procédé de préparation et les compositions pharmaceutiques les contenant. Brevet français N°02/04036, 29/03/2002, 2002.
Capet, M.; Coquerel, G.; Danvy, D.; Lecomte, J.-M.; Petit, M.-N.; Schwartz, J. C.
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2000
Nouvelle forme cristalline "alpha" du sel de ter-butylamine du perindopril, son procédé de fabrication, et les compositions pharmaceutiques qui la contiennent. Brevet N°00/08793, 06/07/2000, 2000.
Pfeiffer, B.; Ginot, Y.-M.; Coquerel, G.; Beilles, S.Nouvelle forme "béta" du del de ter-butylamine du perindopril, son procédé de préparation, et les compositions pharmaceutiques qui la contiennent. Brevet N° 00/08792, 06/07/2000, 2000.
Pfeiffer, B.; Ginot, Y.-M.; Coquerel, G.; Beilles, S. Nouvelle forme cristalline "gamma" de sel de ter-butylamine du perindopril, son procédé de préparation, et les compositions pharmaceutiques qui la contiennent. Brevet N°00/08791, 06/07/2000, 2000.
Pfeiffer, B.; Ginot, Y.-M.; Coquerel, G.; Beilles, S.
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1997
Method for splitting 1-amino-alcan-2-ol compounds. PCT FR97/02158, 28/11/1997, 1997.
Coquerel, G.; Catroux, L.; Combret, Y.
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1996
Procédé de dédoublement par diastéréoisomères et par cristallisation préférentielle dans la série des 1-amino-alcan-2-ols. PCT N°94/01-107, 22/09/1996, 1996.
Coquerel, G.; Catroux, L.; Combret, Y.
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1994
Procédé de dédoublement (AS3PC) de deux antipodes optiques par entraînement polythermique programmé et auto-ensemencé. PCT N°94/01.107, 22/09/1994, 1994.
Coquerel, G.; Petit, M.-N.; Bouaziz, R.
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1993
Procédé de dédoublement de deux antipodes optiques par entraînement polythermique programmé et auto-ensemencé. Brevet français N°93/11354, 23/09/1993, 1993.
Coquerel, G.; Petit, M.-N.; Bouaziz, R.
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1991
Procédé de dédoublement d'hydantoïnes chirales. PCT 91/00906, 15/11/1991, 1991.
Depernet, D.; Bouaziz, R.; Coquerel, G.; Petit, M.-N.
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1990
Procédé de séparation des énantiomères des 5-aryl-5-alkyl hydantoïnes. Brevet français N°90/11487, 16/11/1990, 1990.
Coquerel, G.; Petit, M.-N.; Bouaziz, R.
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Mis à jour le 11/05/2012
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